Which drug induces bilirubin biotransformation?
A) serotonin
B) epinephrine
C) norepinephrine
D) phenobarbital
E) dopamine
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Indinavir and nelfinavir are protease inhibitors used to treat human immunodeficiency virus. Both drugs are known to inhibit UGT1A1 and OATP1B1,15 but only indinavir is associated with hyperbilirubinemia.
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